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BTSA1

Glpbio
Catalog No:GC39355-50mg CAS No.:314761-14-3 MDLNo: Brand:Glpbio purity: 特性: Purpose:BTSA1 是一種有效的,高親和力和口服活性的 BAX 激活劑,IC50 為 250 nM,EC50 為 144 nM。BTSA1 以高親和力和特異性與 N 末端激活位點結(jié)合,并誘導(dǎo) BAX 發(fā)生構(gòu)象變化,從而導(dǎo)致 BAX 介導(dǎo)的細(xì)胞凋亡。DMSO: 25 mg/mL (58.07 mM)
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